1. Signaling Pathways
  2. Antibody-drug Conjugate/ADC Related
  3. ADC Payload
  4. ADC Payload Inhibitors

ADC Payload Inhibitors

Auristatin

Calicheamicins

Camptothecins

Daunorubicins/Doxorubicins

Duocarmycins

Maytansinoids

Pyrrolobenzodiazepines

Traditional Cytotoxic Agents

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ADC Payload
Product Name Auristatin Calicheamicins Camptothecins Daunorubicins/Doxorubicins Duocarmycins Maytansinoids Pyrrolobenzodiazepines Traditional Cytotoxic Agents Purity
Paclitaxel              
Traditional Cytotoxic Agents
99.97%
Monomethyl auristatin E
Auristatin
              99.98%
DXd    
Camptothecins
          99.30%
SN-38    
Camptothecins
          99.94%
Exatecan mesylate    
Camptothecins
          99.98%
Methotrexate              
Traditional Cytotoxic Agents
99.95%
Exatecan    
Camptothecins
          99.93%
Camptothecin    
Camptothecins
          99.77%
MMAF
Auristatin
              99.97%
Mertansine          
Maytansinoids
    99.80%
α-Amanitin              
Traditional Cytotoxic Agents
99.92%
Daunorubicin hydrochloride      
Daunorubicins/Doxorubicins
        99.67%
Exatecan-d5 mesylate    
Camptothecins
          99.83%
MMAE-d8
Auristatin
              99.29%
Calicheamicin  
Calicheamicins
            98.28%
Exatecan Intermediate 1    
Camptothecins
          99.99%
Methotrexate disodium              
Traditional Cytotoxic Agents
99.63%
SG3199            
Pyrrolobenzodiazepines
  98.33%
PNU-159682      
Daunorubicins/Doxorubicins
        98.50%
Exatecan Intermediate 2    
Camptothecins
          99.99%
Daunorubicin      
Daunorubicins/Doxorubicins
        99.94%
(4-NH2)-Exatecan    
Camptothecins
          99.93%
Auristatin E
Auristatin
              99.86%
Exatecan mesylate (GMP)    
Camptothecins
         
Exatecan Intermediate 6    
Camptothecins
          98.98%
Duocarmycin DM free base      
Daunorubicins/Doxorubicins
        99.69%
7-MAD-MDCPT    
Camptothecins
          98.80%
Cyclopropaneacetamide-Exatecan    
Camptothecins
          99.60%
Ansamitocin P-3          
Maytansinoids
    98.0%
PF-06380101
Auristatin
              99.95%
MMAF-OMe
Auristatin
              99.62%
SJG-136            
Pyrrolobenzodiazepines
  99.47%
(αR)-Cyclopropaneacetamide-Exatecan    
Camptothecins
          99.93%
MMAF hydrochloride
Auristatin
              99.97%
Ac-Exatecan    
Camptothecins
          99.02%
β-Amanitin              
Traditional Cytotoxic Agents
98.02%
SG2057            
Pyrrolobenzodiazepines
  99.93%
Duocarmycin TM        
Duocarmycins
      99.82%
(R)-Exatecan Intermediate 1    
Camptothecins
          99.95%
Duocarmycin SA        
Duocarmycins
      99.89%
Daun02      
Daunorubicins/Doxorubicins
        98.72%
γ-Amanitin              
Traditional Cytotoxic Agents
Taltobulin              
Traditional Cytotoxic Agents
99.90%
Tubulysin A              
Traditional Cytotoxic Agents
99.56%
Dolastatin 10
Auristatin
              98.34%
Hemiasterlin            
Pyrrolobenzodiazepines
  99.90%
N-Me-L-Ala-maytansinol          
Maytansinoids
    99.89%
Fmoc-MMAE
Auristatin
              99.35%
Exatecan Intermediate 5    
Camptothecins
          99.98%
MMAD
Auristatin
              99.92%
MMAF sodium
Auristatin
              99.59%
DM4-SMe          
Maytansinoids
    99.99%
DM1-SMe          
Maytansinoids
    99.08%
Glucocorticoid receptor agonist-5              
Traditional Cytotoxic Agents
99.95%
DC0-NH2        
Duocarmycins
     
Duocarmycin GA        
Duocarmycins
      99.00%
Exatecan intermediate 9    
Camptothecins
          99.80%
10-Deacetyl-7-xylosyl paclitaxel              
Traditional Cytotoxic Agents
99.40%
(rac)-Exatecan Intermediate 1    
Camptothecins
          99.97%
Exatecan Intermediate 4    
Camptothecins
          98.95%
MMAF-d8 hydrochloride
Auristatin
              99.52%
PF-06380101-d8
Auristatin
              99.27%
Tomaymycin DM            
Pyrrolobenzodiazepines
 
Exatecan intermediate 10    
Camptothecins
          99.91%
Exatecan Intermediate 2 hydrochloride    
Camptothecins
          99.94%
Exatecan Intermediate 3    
Camptothecins
          99.83%
Exatecan Intermediate 7    
Camptothecins
         
DM3          
Maytansinoids
   
Exatecan-methylacetamide-OH    
Camptothecins
         
Exatecan-amide-cyclopropanol    
Camptothecins
          98.57%
PNU-159682 carboxylic acid      
Daunorubicins/Doxorubicins
       
Exatecan Intermediate 4 dihydrochloride    
Camptothecins
          99.92%
Exatecan analog 36    
Camptothecins
          98.71%
Doxorubicin hydrochloride      
Daunorubicins/Doxorubicins
        99.90%
Doxorubicin      
Daunorubicins/Doxorubicins
       
DC1SMe        
Duocarmycins
      98.0%
Duocarmycin DM      
Daunorubicins/Doxorubicins
        99.15%
Duocarmycin analog-1        
Duocarmycins
     
Maytansinoid DM4          
Maytansinoids
   
(5-Cl)-Exatecan    
Camptothecins
         
Decyclohexanamine-Exatecan    
Camptothecins
          98.92%
S-methyl DM1          
Maytansinoids
    99.58%
Taltobulin hydrochloride              
Traditional Cytotoxic Agents
99.34%
Taltobulin trifluoroacetate              
Traditional Cytotoxic Agents
99.08%
Exatecan mesylate dihydrate    
Camptothecins
         
C-11              
Traditional Cytotoxic Agents
DC1        
Duocarmycins
     
(+)-CBI-CDPI1        
Duocarmycins
     
DM3-SMe          
Maytansinoids
   
DMEA-PNU-159682      
Daunorubicins/Doxorubicins
       
DC41SMe        
Duocarmycins
     
(+)-CBI-CDPI2        
Duocarmycins
     
Duocarmycin MB        
Duocarmycins
     
DC41        
Duocarmycins
     
DC4SMe        
Duocarmycins
     
Seco-Duocarmycin TM        
Duocarmycins
     
Methotrexate monohydrate              
Traditional Cytotoxic Agents
Aniline-MPB-amino-C3-PBD            
Pyrrolobenzodiazepines
 
Rebeccamycin              
Traditional Cytotoxic Agents
DC10SMe        
Duocarmycins
     
Daunorubicin citrate      
Daunorubicins/Doxorubicins
       
Dolastatin 15
Auristatin
             
Isofistularin-3              
Traditional Cytotoxic Agents
Seco-Duocarmycin SA        
Duocarmycins
     
ε-Amanitin              
Traditional Cytotoxic Agents
Gly-Cyclopropane-Exatecan    
Camptothecins
         
Mensacarcin              
Traditional Cytotoxic Agents
Tubulysin IM-2              
Traditional Cytotoxic Agents
Duocarmycin A        
Duocarmycins
     
Py-MPB-amino-C3-PBD            
Pyrrolobenzodiazepines
 
Dimethyl-SGD-1882            
Pyrrolobenzodiazepines
 
Top1 inhibitor 1    
Camptothecins
          99.67%
Exatecan-amide-bicyclo[1.1.1]pentan-1-ylmethanol    
Camptothecins
         
Tubulysin IM-3              
Traditional Cytotoxic Agents
Exatecan-amide-bicyclo[1.1.1]pentan-1-ol    
Camptothecins
         
MMAD-d8
Auristatin
              98.95%
17-AEP-GA              
Traditional Cytotoxic Agents
Polyketomycin              
Traditional Cytotoxic Agents
Azonafide-PEABA              
Traditional Cytotoxic Agents
(1-OH)-Exatecan    
Camptothecins
         
Duocarmycin MA        
Duocarmycins
     
17-GMB-APA-GA              
Traditional Cytotoxic Agents
Exatecan analogue 1    
Camptothecins
         
NH2-methylpropanamide-Exatecan TFA    
Camptothecins
          99.80%
Tubulysin IM-1              
Traditional Cytotoxic Agents
Corixetan              
Traditional Cytotoxic Agents
Sandramycin              
Traditional Cytotoxic Agents
Exatecan intermediate 11    
Camptothecins
         
Exatecan intermediate 8    
Camptothecins
         
Exatecan-amide-CH2-O-CH2-CH2-OH    
Camptothecins